CA2900855C - Aminopyrimidinyl compounds - Google Patents

Aminopyrimidinyl compounds Download PDF

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Publication number
CA2900855C
CA2900855C CA2900855A CA2900855A CA2900855C CA 2900855 C CA2900855 C CA 2900855C CA 2900855 A CA2900855 A CA 2900855A CA 2900855 A CA2900855 A CA 2900855A CA 2900855 C CA2900855 C CA 2900855C
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Canada
Prior art keywords
alkyl
diazabicyclo
pyrimidin
amino
oct
Prior art date
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CA2900855A
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English (en)
French (fr)
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CA2900855A1 (en
Inventor
Andrew Fensome
Ariamala Gopalsamy
Brian S. GERSTENBERGER
Ivan Viktorovich Efremov
Zhao-Kui Wan
Betsy PIERCE
Jean-Baptiste Telliez
John I. Trujillo
Liying Zhang
Li Xing
Eddine Saiah
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Pfizer Corp SRL
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Pfizer Corp SRL
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Application filed by Pfizer Corp SRL filed Critical Pfizer Corp SRL
Publication of CA2900855A1 publication Critical patent/CA2900855A1/en
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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CA2900855A 2014-08-21 2015-08-18 Aminopyrimidinyl compounds Active CA2900855C (en)

Applications Claiming Priority (2)

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US201462039969P 2014-08-21 2014-08-21
US62/039,969 2014-08-21

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CA2900855A1 CA2900855A1 (en) 2016-02-21
CA2900855C true CA2900855C (en) 2022-03-15

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US (5) US9663526B2 (en])
EP (1) EP3183247B9 (en])
JP (1) JP6218260B2 (en])
KR (1) KR101877189B1 (en])
CN (1) CN107074867B (en])
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